Bioactive Compounds
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B5820 RO5126766(CH5126766)Summary: Raf/MEK dual inhibitor -
A8716 LY3009120Target: RafSummary: pan-RAF and RAF dimer inhibitor -
B6088 EPZ020411Summary: PRMT6 inhibitor -
C3171 CBL0137Summary: curaxin that activates p53 and inhibits NF-κB -
C3528 CitrininSummary: mycotoxin that induces apoptosis and blocks tubulin polymerization as well as mitotic spindle assembly -
C4097 NI-57Summary: bromodomains of BRPF proteins inhibitor -
C4226 Phomopsin ASummary: cyclic hexapeptide mycotoxin that binds β-tubulin -
C5478 NCT-502Summary: inhibitor of 3-phosphoglycerate dehydrogenase (PHGDH) -
B1047 GDC-0032Target: PI3KSummary: PI3Kα inhibitor -
B1569 Bepotastine Besilate1 CitationSummary: Non-sedating, selective antagonist of histamine 1 (H1) receptor
