Bioactive Compounds
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B4950 Darunavir EthanolateSummary: nonpeptidic HIV protease inhibitor -
A8702 MesoridazineSummary: A dopaminergic antagonist -
B5998 GSK2801Summary: inhibitor of BAZ2A and BAZ2B bromodomains -
A5760 KRN 633Summary: VEGFR inhibitor,ATP-competitive -
A8335 Palbociclib (PD0332991) Isethionate1 CitationTarget: Cyclin-Dependent KinasesSummary: CDK4/6 inhibitor,highly selective -
A8437 Gemcitabine9 CitationSummary: inhibitor of DNA synthesis -
A8600 Tankyrase Inhibitors (TNKS) 22Summary: Tankyrase inhibitor -
B2184 GDC-0980 (RG7422)Summary: Class I PI3K inhibitor for PI3Kα/β/δ/γ -
B1621 TAK-733Target: MEKSummary: MEK allosteric site inhibitor -
B1303 Amsacrine hydrochlorideSummary: Topoisomerase 2 inhibitor

