Bioactive Compounds
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A4498 SBHA1 CitationTarget: Histone Deacetylases (HDACs)Summary: HDAC1/HDAC3 inhibitor,cell-permeable -
A5181 LinezolidSummary: Antibacterial reagent -
A5294 Sumatriptan SuccinateTarget: 5-HT1 ReceptorsSummary: 5-HT1 receptor agonist -
A8366 ARRY-380Target: HER2Summary: Tyrosine kinase HER2 and p95-HER2 inhibitor -
A8370 Axitinib (AG 013736)5 CitationTarget: VEGFR|PDGFR|c-KitSummary: VEGFR1/ c-Kit inhibitor -
A8505 PKI-402Summary: PI3K inhibitor,selective, reversible and ATP-competitive -
A8379 Betamethasone ValerateSummary: anti-inflammatory corticosteroid -
A8642 R5472 CitationTarget: Cyclin-Dependent KinasesSummary: CDK1/2/4 inhibitor,ATP-competitive -
B3238 XCT790Target: Estrogen and Related ReceptorsSummary: ERRα agonist -
B3246 R788 disodium hexahydrateSummary: potent Syk inhibitor

