Bioactive Compounds
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B7485 ReversanSummary: inhibitor of multidrug resistance-associated protein 1 (MRP1) and P-glycoprotein (P-gp) -
B7623 NPEC-caged-D-AP5Summary: NMDA receptor antagonist -
B7749 KRCA 0008Summary: Ack1 and anaplastic lymphoma kinase (ALK) dual inhibitor -
B5001 H-9 dihydrochlorideSummary: A protein kinase inhibitor that inhibits PKA activity and interferes with EGF signaling. -
B5004 FCCP8 CitationSummary: uncoupler of oxidative phosphorylation -
B5019 7-NINASummary: non-selective NOS inhibitor -
A3004 Vemurafenib (PLX4032, RG7204)13 CitationTarget: RafSummary: BRAF kinase inhibitor -
A3006 GDC-0068 (RG7440)3 CitationTarget: AktSummary: Pan-AKT inhibitor,highly selective -
A3011 CHIR-99021 (CT99021)32 CitationTarget: GSK-3Summary: GSK-3 inhibitor -
A3021 GDC-0449 (Vismodegib)12 CitationTarget: P-glycoprotein (P-gp)|HedgehogSummary: Hedgehog antagonist,potent and selective

