Bioactive Compounds
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A4184 PFI-1 (PF-6405761)1 CitationTarget: BromodomainsSummary: BET inhibitor -
A4110 MLN8237 (Alisertib)12 CitationSummary: Aurora A Kinase inhibitor, Potent and selective -
A4033 GlimepirideTarget: Inward Rectifier Potassium (Kir) ChannelsSummary: Sulfonylurea compound -
A4050 GM 60017 CitationTarget: MMPSummary: Broad spectrum MMP inhibitor -
A2587 PMSF20 CitationTarget: Serine ProteasesSummary: PMSF -
A4221 YM1552 CitationTarget: SurvivinSummary: Survivin suppressant,apoptosis inhibitor -
A4193 SMI-4aTarget: PimSummary: Potent Pim inhibitor -
A1914 UNC06381 CitationSummary: G9a/GLP HMTase inhibitor, potent and selective -
A4318 AvasimibeTarget: Acyl coenzyme A: cholesterol acyltransferasesSummary: ACAT inhibitor,orally bioavailable -
A4336 Mycophenolate MofetilSummary: IMPDH inhibitor

