Bioactive Compounds
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B8772 CFT8634Summary: An orally active BRD9-targeting degrader for research on tumors such as synovial sarcoma. -
A3016 PLX-47201 CitationTarget: RafSummary: BRAF kinase inhibitor -
A3017 Dasatinib (BMS-354825)14 CitationSummary: Src and Bcr-Abl inhibitor -
A4003 LDN 57444Target: UCHSummary: UCH-L1 inhibitor,reversible competitve -
A2576 E-646 CitationTarget: Cathepsins|Calpains|PapainsSummary: cysteine proteases inhibitor -
A2603 Calpain Inhibitor II, ALLM5 CitationSummary: Calpain inhibitor -
A2578 Clasto-Lactacystin β-lactoneTarget: ProteasomeSummary: Proteasome inhibitor -
A4018 YO-01027 (Dibenzazepine, DBZ)1 CitationSummary: γ-secretase inhibitor -
A4056 AT13387Target: HSP90Summary: Hsp90 inhibitor -
A4182 Resveratrol7 CitationTarget: Sir2-like Family Deacetylases (Sirtuins)|COX|LOX|Adenylyl cyclase|Quinone reductaseSummary: SIRT1 activator
