Bioactive Compounds
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A4190 GSK J4 HCl1 CitationSummary: Inhibitor of H3K27 demethylase JMJD3,potent and cell-permeable -
A2588 PPACK DihydrochlorideSummary: Thrombin inhibitor -
A4227 Tipifarnib (Zarnestra)Summary: Farnesyltransferase inhibitor,potent and specific -
A4240 Abiraterone1 CitationSummary: Potent CYP17 inhibitor -
A1900 PSISummary: Proteasome inhibitor -
A1901 Q-VD-OPh88 CitationTarget: CaspasesSummary: pan-caspase inhibitor -
A1903 E 64d9 CitationSummary: Cysteine protease inhibitor -
A1906 Decitabine (NSC127716, 5AZA-CdR)6 CitationSummary: A DNMT1 inhibitor -
A4338 RivaroxabanTarget: Factor XaSummary: Factor Xa inhibitor -
A4345 MK-8245Summary: SCD inhibitor,potent and liver-selective

