Bioactive Compounds
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A4058 BIIB021Target: HSP90Summary: Hsp90 inhibitor,selective and competitive -
A4153 BMN 6737 CitationSummary: Potent PARP inhibitor -
A2583 Lactacystin (Synthetic)1 CitationTarget: ProteasomeSummary: Proteasome inhibitor -
A4072 MK-2048Summary: Integrase inhibitor for HIV-1,second generation -
A4166 EPZ56762 CitationTarget: DOT1LSummary: DOT1L inhibitor,potent and SAM competitive -
A4111 VX-680 (MK-0457,Tozasertib)1 CitationTarget: Aurora KinasesSummary: Aurora kinase inhibitor -
A4034 Linagliptin (BI-1356)Summary: DDP-4 inhibitor,highly potent and competitive -
A2585 MG-132136 CitationTarget: ProteasomeSummary: proteasome inhibitor -
A4051 NSC 4050201 CitationTarget: MMPSummary: MT1-MMP inhibitor -
A4209 NSC 207895 (XI-006)Target: MDMXSummary: MDMX inhibitor,anti-cancer agent
