Bioactive Compounds
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B6208 Dihydrokainic acidSummary: EAAT2(GLT1)-selective non-transportable inhibitor of L-glutamate and L-aspartate uptake -
B7228 CI 1020Summary: endothelin-A receptor (ETA) antagonist -
B7791 6-Bnz-cAMP sodium saltSummary: cAMP analog,PKA activator -
A8902 6H05Summary: K-Ras inhibitor -
A9502 OTS964 hydrochloride1 CitationSummary: TOPK inhibitor,potent and selective -
B4888 Obeticholic Acid2 CitationTarget: Farnesoid X receptors (FXRs)Summary: FXR agonist with anticholeretic activity -
B4889 Verdinexor (KPT-335)Summary: XPO1/CRM1 inhibitor -
B4900 Indoximod (NLG-8189)Summary: Indoleamine 2,3-dioxygenase (IDO) pathway inhibitor -
B4924 TA 02Summary: p38 MAPK inhibitor -
B4932 JJKK 048Summary: monoacylglycerol lipase (MAGL) inhibitor

