Bioactive Compounds
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B7679 (R)-(+)-Etomoxir sodium saltSummary: carnitine palmitoyltransferase I (CPT1) inhibitor -
B5086 CGP 55845 hydrochloride2 CitationTarget: GABAB ReceptorsSummary: GABAB receptor antagonist -
A4007 MLN9708 Analogue6 CitationTarget: ProteasomeSummary: Proteasome inhibitor -
A4093 ITF2357 (Givinostat)2 CitationTarget: Histone Deacetylases (HDACs)Summary: HDAC inhibitor -
A4065 PF-04929113 (SNX-5422)Target: HSP90Summary: Hsp90 inhibitor,potent and selective -
A4160 A-966492Target: PARPSummary: PARP-1/-2 inhibitor, highly potent -
A4117 AT9283Summary: Aurora kinase/JAK inhibitor -
A4217 QNZ (EVP4593)6 CitationSummary: Potent NF-κB inhibitor -
A4305 WY-14643 (Pirinixic Acid)10 CitationTarget: PPARSummary: PPARα agonist,selective and highly potent -
A4327 TadalafilTarget: Phosphodiesterases (PDEs)Summary: PDE5 inhibitor

