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Ketoconazole

Catalog No.
A4316
Inhibitor of cyclosporine oxidase and testosterone 6 beta-hydroxylase
Grouped product items
SizePriceStock Qty
10mM (in 1mL DMSO)
$80.00
In stock
500mg
$65.00
In stock

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Email: [email protected]

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Background

Ketoconazole inhibits cyclosporine oxidase and testosterone 6 beta-hydroxylase with IC50 of 0.19 mM and 0.22 mM, respectively.

Chemical Properties

Physical AppearanceA solid
StorageStore at -20°C
M.Wt531.43
Cas No.65277-42-1
FormulaC26H28Cl2N4O4
Solubility≥23.4 mg/mL in DMSO, ≥10 mg/mL in EtOH with ultrasonic,insoluble in H2O
Chemical Name1-[4-[4-[[(2R,4S)-2-(2,4-dichlorophenyl)-2-(imidazol-1-ylmethyl)-1,3-dioxolan-4-yl]methoxy]phenyl]piperazin-1-yl]ethanone
SDFDownload SDF
Canonical SMILESCC(=O)N1CCN(CC1)C2=CC=C(C=C2)OCC3COC(O3)(CN4C=CN=C4)C5=C(C=C(C=C5)Cl)Cl
Shipping ConditionEvaluation sample solution : ship with blue ice.All other available size: ship with RT , or blue ice upon request
General tipsFor obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20℃ for several months.

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