EGFR
EGFR (epidermal growth factor receptor) is the cell-surface receptor of its specific ligands, including epidermal growth factor and TGFα (transforming growth factor α) and is a receptor tyrosine kinase.
- A4139 AG-4903 CitationTarget: EGFR|JAKSummary: JAK2/EGFR inhibitor
- A3256 BMS-690514Summary: HER/EGFR inhibitor
- A3320 CO-1686 (AVL-301)1 CitationTarget: EGFRSummary: EGFR inhibitor
- A3397 Erlotinib4 CitationSummary: EGFR tyrosine kinase inhibitor
- A3433 Gefitinib hydrochlorideTarget: EGFRSummary: Potent EGFR inhibitor
- A3482 Icotinib HydrochlorideSummary: EGFR inhibitor,potent and specific
- A3967 Lapatinib DitosylateTarget: EGFR|ErbB-2Summary: EGFR/HER2 inhibitor,potent and selective
- A8218 Lapatinib7 CitationTarget: ErbBSummary: EGFR/HER2 inhibitor,potent,selective and reversible
- A8219 Gefitinib (ZD1839)15 CitationTarget: EGFRSummary: Selective EGFR inhibitor
- A8234 Erlotinib Hydrochloride2 CitationSummary: Selective EGFR inhibitor