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Trelagliptin succinate

Catalog No.
A3889
DPP-4 inhibitor
Grouped product items
SizePriceStock Qty
5mg
$113.00
Ship with 10-15 days
10mg
$180.00
Ship with 10-15 days
50mg
$720.00
Ship with 10-15 days
100mg
$1,215.00
Ship with 10-15 days

Tel: +1-832-696-8203

Email: [email protected]

Worldwide Distributors

Background

Trelagliptin is a long acting dipeptidyl peptidase-4 (DPP-4) inhibitor that is being developed for the treatment of type 2 diabetes (T2D). Two Phase II clinical studies have been completed with Efficacy and Safety of SYR-472 in Subjects With Type 2 Diabetes Mellitus. Phase III clinical studies with trelagliptin in Japan to evaluate its safety and efficacy in a once-weekly oral treatment regimen. Currently, all available DPP-4 inhibitors are dosed once-daily. A once-weekly treatment, such as trelagliptin, would provide patients with a convenient treatment alternative and has the potential to improve treatment compliance.

Chemical Properties

StorageStore at -20°C
M.Wt475.47
Cas No.1029877-94-8
FormulaC22H26FN5O6
SynonymsSYR-472 succinate;SYR472 succinate;SYR 472 succinate
SolubilitySoluble in DMSO
Chemical Name2-[[6-[(3R)-3-aminopiperidin-1-yl]-3-methyl-2,4-dioxopyrimidin-1-yl]methyl]-4-fluorobenzonitrile;butanedioic acid
SDFDownload SDF
Canonical SMILESCN1C(=O)C=C(N(C1=O)CC2=C(C=CC(=C2)F)C#N)N3CCCC(C3)N.C(CC(=O)O)C(=O)O
Shipping ConditionEvaluation sample solution : ship with blue ice.All other available size: ship with RT , or blue ice upon request
General tipsFor obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20℃ for several months.

Quality Control

Quality Control & MSDS

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Chemical structure

Trelagliptin succinate