Cyclin-Dependent Kinases
Cyclin-dependent kinases is a group of serine/threonine kinases. It is activated by binding to cyclin and participates in the regulation of cell cycle.
- B3277 AMG 925Target: Cyclin-Dependent Kinases|FLT3Summary: FLT3/CDK4 inhibitor,potent and selective
- B4754 LDC0000672 CitationTarget: Cyclin-Dependent KinasesSummary: CDK9 inhibitor, novel and highly specific
- B8002 LY2857785Summary: CDK9 inhibitor
- A8885 Ro 33064 CitationTarget: Cyclin-Dependent KinasesSummary: An ATP-competitive, potent CDK1 inhibitor
- B4990 Purvalanol ASummary: potent, and cell-permeable CDK inhibitor
- B5926 AZD-5597Summary: Potent CDK inhibitor
- A8717 THZ21 CitationTarget: Cyclin-Dependent KinasesSummary: CDK7 inhibitor
- A8718 GX-674Target: Voltage-gated Sodium (NaV) ChannelsSummary: Nav1.7 antagonist
- B6042 K03861Summary: CDK2 inhibitor
- A8736 THZ531Target: Cyclin-Dependent KinasesSummary: CDK12 and CDK13 covalent inhibitor