Signaling Pathways
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A4545 TCS 401Summary: Selective PTP1B inhibitor -
A4548 α-Amanitin10 CitationSummary: RNA polymerase II inhibitor -
A4453 NSC 687852 (b-AP15)Target: Deubiquitinating enzymes (DUBs)Summary: 19S regulatory particle Inhibitor -
A4477 Cyclic Pifithrin-α hydrobromideSummary: P53 inhibitor -
A4482 Pifithrin-μ1 CitationTarget: Autophagy|p53|HSP70Summary: Inhibitor of p53 binding and anti-apoptotic -
A4484 PRIMA-1METSummary: Restore mutant p53 activity, induce BAX and PUMA -
A3963 A-7696624 CitationSummary: AMPK activator,potent and reversible -
A3965 BI 25361 CitationTarget: PLK|Bromodomain-containing proteins(BRDs)Summary: Plk1 inhibitor,potent and ATP-competitive -
A3966 Doxorubicin3 CitationSummary: DNA topoisomerase II inhibitor -
A3967 Lapatinib DitosylateTarget: EGFR|ErbB-2Summary: EGFR/HER2 inhibitor,potent and selective

