T025
Catalog No.
BA2818
T025 is an orally effective inhibitor.
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T025 is an orally potent inhibitor of CLK1, CLK2, CLK3, CLK4, DYRK1A, DYRK1B, and DYRK2 at 4.8, 0.096, 6.5, 0.61, 0.074, 1.5, and 32 nM, respectively.T025 induces caspase-3/7-mediated apoptosis.T025 reduces the dependence phosphorylation T025 has antiproliferative activity in both hematological and solid cancer cell lines (IC: 30-300nM).T025 has antitumor efficacy and is mainly used in MYC-driven disease research.
| Physical Appearance | A solid |
| Storage | -20°C |
| M.Wt | 382.42 |
| Cas No. | 2407433-00-3 |
| Formula | C21H18N8 |
| Chemical Name | N2-methyl-N4-(pyrimidin-2-ylmethyl)-5-(quinolin-6-yl)-7H-pyrrolo[2,3-d]pyrimidine-2,4-diamine |
| Canonical SMILES | CNC1=NC(NCC2=NC=CC=N2)=C3C(C4=CC=C5C(C=CC=N5)=C4)=CNC3=N1 |
| Shipping Condition | Small Molecules with Blue Ice, Modified Nucleotides with Dry Ice. |
| General tips | We do not recommend long-term storage for the solution, please use it up soon. |
Quality Control & MSDS
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Chemical structure
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