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Cercosporamide

Catalog No.
A4511
Mnk2 and JAK3 inhibitor
Grouped product items
SizePriceStock Qty
500ug
$894.00
Ship with 10-15 days
1mg
$1,481.00
Ship with 10-15 days
For scientific research use only and should not be used for diagnostic or medical purposes.

Tel: +1-832-696-8203

Email: [email protected]

Worldwide Distributors

Background

Potent inhibitor of MAP-kinase interacting kinase-2 (Mnk2) and JAK3 (IC50 values are 11, 31 and 116 nM for Mnk2, JAK3 and Mnk1 respectively). Blocks eIF4E phosphorylation; exhibits antiproliferative and proapoptotic activity in cancer cells in vitro. Also inhibits Pkc1. Orally bioavailable.

Chemical Properties

Physical AppearanceA light to dark tan solid
StorageStore at -20°C
M.Wt331.28
Cas No.131436-22-1
FormulaC16H13NO7
SolubilityLimited solubility, soluble in DMSO
Chemical Name(9aS)-8-acetyl-1,3,7-trihydroxy-9a-methyl-9-oxodibenzofuran-4-carboxamide
SDFDownload SDF
Canonical SMILESC[C@@](C(Oc1c(C(N)=O)c(O)c2)=CC(O)=C3C(C)=O)(c1c2O)C3=O
Shipping ConditionSmall Molecules with Blue Ice, Modified Nucleotides with Dry Ice.
General tips We do not recommend long-term storage for the solution, please use it up soon.

Quality Control

Quality Control & MSDS

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Chemical structure

Cercosporamide