BMS-470539 dihydrochloride
Catalog No.
A9969
A highly selective melanocortin 1 receptor (MC-1R) agonist
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BMS-470539 dihydrochloride is a highly selective melanocortin 1 receptor (MC-1R) agonist, with an IC50 value of 120 nM and an EC50 value of 28 nM, indicating high affinity and agonist activity for MC-1R. Melanocortin 1 receptor (MC-1R) is widely found in skin melanocytes and is involved in regulating the physiological processes of melanin synthesis, skin pigmentation and anti-inflammatory response. BMS-470539 dihydrochloride promotes melanin generation effectively by selectively activating MC-1R, which has potential application prospects for the treatment of skin pigmentation disorders.
| Storage | Store at -20°C for 3 years. |
| M.Wt | 632.63 |
| Cas No. | 2341796-82-3 |
| Formula | C32H43Cl2N5O4 |
| Solubility | Soluble in DMSO |
| Chemical Name | (S)-2-amino-N-((R)-1-(4-butyryl-4-phenylpiperidin-1-yl)-3-(4-methoxyphenyl)-1-oxopropan-2-yl)-3-(1-methyl-1H-imidazol-5-yl)propanamide dihydrochloride |
| SDF | Download SDF |
| Canonical SMILES | N[C@@H](CC1=CN=CN1C)C(N[C@@H](C(N2CCC(C3=CC=CC=C3)(C(CCC)=O)CC2)=O)CC4=CC=C(OC)C=C4)=O.Cl.Cl |
| Shipping Condition | Small Molecules with Blue Ice, Modified Nucleotides with Dry Ice. |
| General tips | We do not recommend long-term storage for the solution, please use it up soon. |
Quality Control & MSDS
- View current batch:
-
Purity = 98.00%
- COA (Certificate Of Analysis)
- MSDS (Material Safety Data Sheet)
Chemical structure
