Tianeptine
Catalog No.
A3873
5-HT facilitator
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Tianeptine is a selective facilitator of 5-HT uptake in vitro and in vivo. Tianeptine has no affinity for a wide range of receptors, including 5-HT and dopamine (IC50 > 10 μM) and has no effect on noradrenalin or dopamine uptake. Antidepressant, analgesic and neuroprotective following systemic administration in vivo.
| Storage | Store at -20°C |
| M.Wt | 436.96 |
| Cas No. | 72797-41-2 |
| Formula | C21H25ClN2O4S |
| Synonyms | Coaxil |
| Solubility | insoluble in H2O; ≥4.08 mg/mL in EtOH with gentle warming and ultrasonic; ≥82.4 mg/mL in DMSO |
| Chemical Name | 7-[(3-chloro-6-methyl-5,5-dioxo-11H-benzo[c][2,1]benzothiazepin-11-yl)amino]heptanoic acid |
| SDF | Download SDF |
| Canonical SMILES | CN(c1ccccc1C(c(cc1)c2cc1Cl)NCCCCCCC(O)=O)S2(=O)=O |
| Shipping Condition | Small Molecules with Blue Ice, Modified Nucleotides with Dry Ice. |
| General tips | We do not recommend long-term storage for the solution, please use it up soon. |
Quality Control & MSDS
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Chemical structure










