Relutrigine
Catalog No.
BA6980
Relutrigine (PRAX-562) is an orally active, persistent sodium channel inhibitor.
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Relutrigine (PRAX-562) is an orally active, persistent sodium channel inhibitor.Relutrigine potently and preferentially inhibits persistent I induced by ATX-II (Nav1.5 activator) or the SCN8A mutation N1768D, with values of 141nM and 75nM, respectively.Relutrigine exhibits use dependent blockade that reduced intrinsic neuronal excitability.Relutrigine has potent anticonvulsant activity.
Physical Appearance | A solid |
Storage | -20°C |
M.Wt | 407.27 |
Cas No. | 2392951-29-8 |
Formula | C15H11F6N5O2 |
Synonyms | PRAX-562 |
Shipping Condition | Small Molecules with Blue Ice, Modified Nucleotides with Dry Ice. |
General tips | We do not recommend long-term storage for the solution, please use it up soon. |