INCB 3284 dimesylate
Catalog No.
A3492
HCCR2 antagonist
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INCB 3284 is a potent, selective and orally bioavailable hCCR2 antagonist. INCB 3284 exhibits potenct antagonism against monocyte chemoattractant molecule binding to hCCR2 and chemotaxis activity (IC50 values are 3.7 and 4.7 nM respectively). INCB 3284 also displays weak hERG activity; inhibits the hERG potassium current (IC50 = 84μM).
| Physical Appearance | A crystalline solid |
| Storage | Store at -20°C |
| M.Wt | 712.76 |
| Cas No. | 887401-93-6 |
| Formula | C28H39F3N4O10S2 |
| Synonyms | INCB-3284 dimesylate;INCB3284 dimesylate |
| Solubility | Soluble in DMSO |
| Chemical Name | N-(2-((1-(4-hydroxy-4-(6-methoxypyridin-3-yl)cyclohexyl)pyrrolidin-3-yl)amino)-2-oxoethyl)-3-(trifluoromethyl)benzamide dimethanesulfonate |
| SDF | Download SDF |
| Canonical SMILES | COC1=NC=C(C2(O)CCC(N3CCC(NC(CNC(C4=CC(C(F)(F)F)=CC=C4)=O)=O)C3)CC2)C=C1.CS(=O)(O)=O.CS(=O)(O)=O |
| Shipping Condition | Small Molecules with Blue Ice, Modified Nucleotides with Dry Ice. |
| General tips | We do not recommend long-term storage for the solution, please use it up soon. |
Quality Control & MSDS
- View current batch:
-
Purity = 98.00%
- COA (Certificate Of Analysis)
- MSDS (Material Safety Data Sheet)
Chemical structure
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