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GNA002

Catalog No.
BA4854
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GNA002 is a potent, selective, covalent inhibitor.
Grouped product items
SizePriceStock Qty
1mg
$342.00
Ship with 10-15 days
5mg
$855.00
Ship with 10-15 days
For scientific research use only and should not be used for diagnostic or medical purposes.

Tel: +1-832-696-8203

Email: [email protected]

Worldwide Distributors

Background

GNA002 is a potent, selective, covalent inhibitor that specifically and covalently binds Cys668 within the EZH2-SET domain, triggering degradation via the COOH terminus of the interacting protein (CHIP)-mediated ubiquitination.GNA002 effectively reduces mediated H3K27 trimethylation and reactivates polycomb repression complex 2 (PRC2) silencing of tumor suppressor genes.

Chemical Properties

Physical AppearanceAn oil
Storage-20°C
M.Wt701.89
Cas No.1385035-79-9
FormulaC42H55NO8
Shipping ConditionSmall Molecules with Blue Ice, Modified Nucleotides with Dry Ice.
General tips We do not recommend long-term storage for the solution, please use it up soon.