BI-4020
Catalog No.
BA6333
BI-4020 is a fourth generation, orally active, non-covalent tyrosine kinase inhibitor.
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BI-4020 is a fourth-generation, orally active, non-covalent tyrosine kinase inhibitor.BI-4020 inhibits not only the triple-mutant del19T790MC797S mutant (=0.2nM in the BaF3 cell line), but also the double-mutant del19T790M and the single-mutant del19 (=1nM).BI-4020 also retained activity against wt (=190nM).BI-4020 showed high kinome selectivity and good DMPK properties.
| Physical Appearance | A solid |
| Storage | -20°C |
| M.Wt | 542.68 |
| Cas No. | 2664214-60-0 |
| Formula | C30H38N8O2 |
| Shipping Condition | Small Molecules with Blue Ice, Modified Nucleotides with Dry Ice. |
| General tips | We do not recommend long-term storage for the solution, please use it up soon. |