Signaling pathways
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BA4379 NMS-P515Summary: NMS-P515 is a potent, orally effective, stereotactic inhibitor. -
BA4380 MSC2504877Summary: MSC2504877 (M2912) is a potent, orally active inhibitor with IC values of 0.0007, 0.0008, and 0.54 μM for TNKS, TNKS2, and PARP1, respectively. -
BA4381 5-AIQSummary: 5-AIQ (5-Aminoisoquinolin-1-one) is a water-soluble inhibitor. -
BA4382 PARP-1-IN-4Summary: PARP-1-IN-4 is an inhibitor. -
BA4383 ART-IN-1Summary: An inhibitor. -
BA4384 PARP1-IN-11Summary: PARP1-IN-11 is a potent inhibitor. -
BA4385 2-Methylquinazolin-4-olSummary: 2-Methylquinazolin-4-ol is a potent, competitive inhibitor. -
BA4386 PARP1-IN-7Summary: PARP1-IN-7 is an inhibitor. -
BA4387 Tankyrase-IN-2Summary: Tankyrase-IN-2 is a potent and selective inhibitor (values of 10 nM, 7 nM, and 710 nM for TNKS1, TNKS2, respectively). -
BA4388 AmelparibSummary: Amelparib is a potent, orally active, water-soluble inhibitor.

