Signaling pathways
- BA5478 ONO-0300302Summary: ONO-0300302 is an orally effective (lysophosphatidic acid receptor 1) antagonist.
- BA5479 NAEPASummary: NAEPA is a phosphate mimetic derivative.
- BA5480 VibozilimodSummary: Agonists.
- BA5481 ZectivimodSummary: Zectivimod is a sphingosine 1-phosphate receptor agonist.
- BA5482 Ex26Summary: Ex26 (S1P1-IN-Ex26) is a potent and selective antagonist (=0.93 nM) with approximately 3,000-fold greater selectivity for S1P than other Sphingosine1-phosphatereceptors.
- BA5483 PCS1055Summary: PCS1055 is a selective and competitive muscarinic-type M4 receptor antagonist.
- BA5484 XanomelineSummary: Xanomeline increases neuronal excitability as a potent selective muscarinic type 1 and type 4 receptor agonist.
- BA5485 PilocarpineSummary: A selective M3 muscarinic acetylcholine receptor agonist.
- BA5487 EmraclidineSummary: Emraclidine (CVL-231) is a modulator (WO2018002760, compound 11).
- BA5488 IperoxoSummary: Iperoxo is a potent super agonist of muscarinic acetylcholine receptors.