Signaling pathways
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BA4998 LP-211Summary: LP-211 is a selective, receptor agonist that crosses the blood-brain barrier. - BA4999 LevomepromazineSummary: Levomepromazine (Methotrimeprazine) is an orally effective antipsychotic active molecule commonly used to relieve nausea and vomiting.
- BA5001 NefazodoneSummary: Nefazodone is an orally active phenylpiperazine antidepressant.
- BA5002 TG6-10-1Summary: An antagonist that acts effectively at low nanomolar levels on EP2, with 300-fold higher selectivity for human EP3, EP4 and IP receptors and 100-fold higher selectivity for EP1 receptors.
- BA5003 2-Methyl-5-HTSummary: 2-Methyl-5-HT (2-Methyl-5-hydroxytryptamine) is a potent and selective agonist.
- BA5004 SarizotanSummary: Sarizotan (EMD128130) is an agonist with oral activity.
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BA5006 GepironeSummary: Gepirone is a selective, affinity agonist. - BA5007 PhenylbiguanideSummary: Phenylbiguanide is a selective receptor agonist.
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BA5009 Perospirone1 CitationSummary: Perospirone (SM-9018freebase) is an orally active antagonist of the receptor (=0.6nM) and receptor (=1.4nM) and a partial agonist of the receptor (=2.9nM). - BA5010 F-15599Summary: F-15599 is a highly selective agonist.