Signaling pathways
- BA5657 6β-NaltrexolSummary: 6β-Naltrexol (6β-Hydroxynaltrexone) is the major metabolite of Naltrexone, a peripherally selective antagonist.
- BA5658 AT-121Summary: AT-121 is a bifunctional and mu opioid receptor agonist.
- BA5659 nor-BinaltorphimineSummary: nor-Binaltorphimine is a selective antagonist.
- BA5660 BMS-986188Summary: S-986188 is a selective orthotropic modulator.
- BA5661 DanavorextonSummary: Danavorexton (TAK-925) is a cerebropermeable agonist of the orexin receptor.
- BA5662 SeltorexantSummary: Seltorexant (JNJ-42847922) is an orally active, high affinity and selective orexin-2 receptor antagonist.
- BA5663 MK-1064Summary: MK-1064 is a selective, orally active antagonist (0.5nM,:18nM).
- BA5664 SB-649868Summary: SB-649868 is an orally effective selective orexin and receptor antagonist.
- BA5665 FirazorextonSummary: Firazorexton (TAK-994freebase) is an orally active, brain-permeable orexin type 2 receptor agonist.
- BA5666 YNT-185Summary: YNT-185 is a non-peptide, selective orexin type 2 receptor agonist.