Signaling pathways
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BA8156 BI-2545Summary: BI-2545 is a potent inhibitor. -
BA8157 EnsifentrineSummary: Ensifentrine (RPL-554) is an inhaled, first-of-its-kind phosphodiesterase 3 and dual inhibitor of 0.4nM and 1479nM, respectively. -
BA8158 PF-05180999Summary: PF-05180999 (PF-999) is a phosphodiesterase 2A inhibitor. -
BA8159 PDE4B-IN-2Summary: PDE4B-IN-2 is an orally active, selective inhibitor. -
BA8160 EurycomanoneSummary: May promote spermatogenesis by inhibiting phosphodiesterase and aromatase activity during estrogen production. -
BA8161 TMX-4100Summary: TMX-4100 is a selective phosphodiesterase 6D degrader. -
BA8162 RoflupramSummary: Roflupram is a selective, orally active inhibitor that crosses the blood-brain barrier. -
BA8163 D159687Summary: An inhibitor. -
BA8164 OrismilastSummary: Orismilast (LEO-32731) is an orally active, selective inhibitor for inflammatory diseases. -
BA8165 PF-05085727Summary: PF-05085727 is a potent cGMP-dependent (=2nM) selective and brain permeable inhibitor.

