Search results for: 'research-area gpcr-g-protein angiotensin-receptor'
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- Target: EGFR|ErbBSummary: ErbB inhibitor
- Target: CSF-1R|VEGFR|PDGFR|c-Kit|FGFRSummary: VEGFR/PDGFR/FGFR inhibitor
- 2 CitationTarget: ErbBSummary: EGFR/HER2 inhibitor,potent,selective and reversible
- Target: PKC|PKG|PKA|Myosin light chain kinases (MLCKs)Summary: protein kinase inhibitor
- Target: CSF-1R|FLT3|VEGFR|PDGFR|c-Kit|FGFRSummary: Oral tyrosine kinase inhibitor (TKI) against FGFR1–3, VEGFR1–3, and platelet-derived growth factor receptor (PDGFR).
- 1 CitationTarget: Vitamin D receptors (VDRs)Summary: Vitamin D receptor activator
- Target: PARSummary: PAR1 agonist
- Target: PARSummary: PAR2 agonist,potent and selective
- Target: Farnesoid X receptors (FXRs)|Vitamin D receptors (VDRs)|Pregnane X receptor(PXR)Summary: Activator of vitamin D receptor,PXR and FXR
- 1 CitationTarget: CSF-1RSummary: CFMS kinase/CSF-1R inhibitor,selective and ATP-competitive