Search results for: 'research-area metabolism'
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- A4383 TolcaponeTarget: Catechol O-Methyltransferase (COMT)Summary: COMT inhibitor
- A4381 FK866 (APO866)1 CitationTarget: NamptSummary: NAMPT inhibitor, non-competitive, highly specific
- A4375 Anacetrapib (MK-0859)1 CitationTarget: CETPSummary: RhCETP/mutant CETP(C13S) inhibitor
- A4367 Atorvastatin CalciumTarget: HMG-CoA ReductasesSummary: HMG-CoA reductase inhibitor
- A4347 Methotrexate2 CitationTarget: Folate AnalogueSummary: Folate antagonist,inhibits DFHR
- A4316 KetoconazoleTarget: Cytochrome P450 (CYP450)Summary: Inhibitor of cyclosporine oxidase and testosterone 6 beta-hydroxylase
- A8202 Abiraterone acetateTarget: Cytochrome P450 (CYP450)Summary: Cytochrome p450 17a1 inhibitor