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GABA Receptor

GABA receptors are a class of receptors that respond to the GABA (neurotransmitter gamma-aminobutyric acid), the chief inhibitory neurotransmitter in the vertebrate central nervous system.


  1. Cat.No. Product Name Information
  2. A3142 Acamprosate calcium GABA receptor agonist and modulator of glutamatergic systems
  3. B1530 Niflumic acid Ca2+-activated Cl- channel blocker
  4. B1532 Nefiracetam GABA receptor activator
  5. B1246 Etomidate hydrochloride GABAA receptors agonist
  6. B2280 Rufinamide voltage-gated sodium channel blocker
  7. B1107 (R)-Baclofen hydrochloride GABAB receptor agonist
  8. B1531 (R)-baclofen GABA receptor agonist
  9. B1024 AWD 131-138 GABAA receptor agonist
  10. A8436 Gabapentin GABA enhancer
  11. A1958 Etomidate General anesthetic with GABA modulatory and GABA-mimetic actions
  12. A2917 Flumazenil Benzodiazepine antagonist
  13. A3917 Vigabatrin GABA transaminase inhibitor
  14. B6914 ZK 93426 hydrochloride benzodiazepine receptor antagonist,competitive
  15. B6915 Ro 15-4513 benzodiazepine ligand
  16. B6918 GS 39783 Positive allosteric modulator of GABAB receptor
  17. B7068 CGS 20625 partial agonist for the benzodiazepine binding site of the GABAA receptor
  18. B7081 (-)-Bicuculline methiodide GABAA receptor antagonist
  19. B7092 Ganaxolone positive allosteric modulator of GABAA receptor
  20. B7151 17-PA GABAA receptor antagonist
  21. B7164 U 90042 GABAA receptor ligand
  22. B7165 U 89843A Positive allosteric modulator of GABAA receptors
  23. B6913 Ro 19-4603 Benzodiazepine inverse agonist
  24. B6912 ZK 93423 hydrochloride GABAA receptor agonist
  25. B6866 N-ArachidonylGABA arachidonyl amino acid
  26. B6677 CI 966 hydrochloride GABA transporter GAT-1 inhibitor
  27. B6692 L-655,708 inverse agonist for the benzodiazepine site of GABAA receptors containing the α5 subunit
  28. B6770 SB 205384 positive GABAA receptor modulator
  29. B6771 CGP 7930 Positive allosteric modulator of GABAB receptors
  30. B6772 CGP 13501 Positive modulator of GABAB receptors,allosteric
  31. B6790 Tracazolate hydrochloride GABAA receptor modulator
  32. B6792 (S)-SNAP 5114 GABA uptake inhibitor
  33. B6840 CL 218872 Benzodiazepine agonist
  34. B6854 NNC 711 GABA uptake inhibitor
  35. B7169 Org 20599 GABAA receptor agonist
  36. B7170 U 93631 GABAA receptor antagonist
  37. B7172 NNC 05-2090 hydrochloride GABA uptake inhibitor
  38. B5482 MRK 016 GABAA receptor inverse agonist
  39. B5499 TCS 1105 GABAA benzodiazepine receptor (BZR) ligand
  40. B5582 Ocinaplon GABAA receptors modulator
  41. B5584 TP 003 GABAA receptor (α3 subtype) partial agonist
  42. B5585 MK 0343 GABAA partial agonist
  43. B5608 PHP 501 trifluoroacetate GABAA antagonist
  44. B6248 Muscimol GABAA receptor agonist, potent
  45. B5646 Pentobarbital sodium salt enhances GABAergic activity
  46. B6102 NS 11394 GABA(A) receptor-positive modulator
  47. B5086 CGP 55845 hydrochloride GABAB receptor antagonist
  48. B5040 SCH 50911 GABAB antagonist
  49. B7214 TB 21007 GABAA receptor inverse agonist
  50. B7253 Alphaxalone activates and potentiates GABAA receptor-activated membrane current (IGABA)
  51. B7268 DMCM hydrochloride Benzodiazepine inverse agonist
  52. B7319 CGP 36216 hydrochloride Selective GABAB antagonist
  53. B7331 L-838,417 Subtype-selective GABAA receptor partial agonist
  54. B7359 rac BHFF GABAB receptor positive allosteric modulator
  55. B7467 DS2 Positive allosteric modulator of δ-subunit containing GABAA receptors
  56. B7544 TCS 1205 GABAA α2 agonist and GABAA α1 partial agonist
  57. B7554 AA 29504 GABAA receptor modulator
  58. C5195 6-(4-Methoxyphenyl)-3-pyridazinamine GABAA receptor antagonist
  59. A3400 Etifoxine GABAA receptor potentiator
  60. B7152 Pentylenetetrazole CNS stimulant
  61. B7254 Valerenic acid Positive allosteric modulator of GABAA receptor
  62. B7430 Bretazenil GABAA benzodiazepine site partial agonist
  63. B7455 Pregnanolone GABAA receptor positive allosteric modulator
  64. B7456 Allopregnanolone GABAA receptor positive allosteric modulator
  65. B5054 Picrotoxin GABAA receptor antagonist
  66. B5356 DPNI-caged-GABA activates GABAA receptor
  67. B5418 RuBi-GABA Ruthenium-bipyridine-triphenylphosphine caged GABA
  68. B5690 RuBi GABA trimethylphosphine GABAB receptor agonist
  69. B6959 Hispidulin Partial positive allosteric modulator at the benzodiazepine receptor
  70. B6953 SCS GABAA receptor antagonist
  71. A3401 Etifoxine hydrochloride GABAA receptor potentiator
  72. A3758 Retigabine dihydrochloride Antiepileptic compound
  73. A3810 SDZ 220-581 Ammonium salt NMDA glutamate receptor antagonist
  74. B6229 Guvacine hydrochloride GABA uptake inhibitor
  75. B6230 Isoguvacine hydrochloride GABAA receptor agonist
  76. B6231 (±)-Nipecotic acid GABA uptake inhibitor
  77. B6327 Dihydroergotoxine mesylate GABAA receptor modulator
  78. B6350 FG 7142 benzodiazepine inverse agonist and anxiogenic agent
  79. B6460 THIP hydrochloride GABAA receptor agonist and GABAA-ρ receptor antagonist
  80. B6207 (-)-Bicuculline methobromide GABAA antagonist
  81. B6210 (-)-Bicuculline methochloride GABAA antagonist
  82. B6216 ZAPA sulfate GABAA receptors agonist
  83. B6487 Chlormethiazole hydrochloride GABAA agonist
  84. B6562 TPMPA GABAA-ρ antagonist
  85. B6589 SKF 89976A hydrochloride GABA uptake inhibitor
  86. B6593 CGP 54626 hydrochloride GABAB receptor antagonist
  87. B6654 CGP 35348 Selective GABAB antagonist, brain penetrant
  88. B6655 CGP 52432 GABAB receptor antagonist
  89. B6656 CGP 46381 GABAB receptor antagonist
  90. B6663 SR 95531 hydrobromide GABAA receptor antagonist
  91. B6676 Loreclezole hydrochloride GABAA receptor modulator
  92. B6450 NCS-382 γ-Hydroxybutyric acid antagonist
  93. B6443 GBLD 345 GABAA receptor agonist
  94. B6401 PK 11195 peripheral benzodiazepine antagonist
  95. B6217 TACA GABAA agonist
  96. B6234 2-Hydroxysaclofen GABAB receptor antagonist
  97. B6235 Saclofen GABAB receptor antagonist
  98. B6282 SKF 97541 GABAB agonist
  99. B6285 3-Methyl-GABA GABA aminotransferase activator
  100. B6291 β-CCB benzodiazepine receptor ligand
  101. B6341 trans-4-Hydroxycrotonic acid ligand of γ-hydroxybutyric acid (GHB) receptor
  102. B6394 FGIN-1-27 high affinity agonist of the translocator protein (TSPO,peripheral benzodiazepine receptor)
  103. B6395 FGIN-1-43 ligand as probe for the mitochondial DBI receptor (peripheral benzodiazepine receptor)
  104. B6215 Phaclofen GABAB antagonist