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TFLLR-NH2

Catalog No.
A8666
PAR1 selective agonist
Grouped product items
SizePriceStock Qty
1mg
$288.00
In stock

Tel: +1-832-696-8203

Email: [email protected]

Worldwide Distributors

Background

Peptide derived from the protease-activated receptor-1 (PAR1) that acts as a PAR1 selective agonist (EC50 = 1.9 μM). Stimulates PAR1-mediated plasma extravasation in vivo. Control Peptide RLLFT-NH2 also available.

Chemical Properties

Physical AppearanceWhite lyophilised solid
StorageDesiccate at -20°C
M.Wt647.82
Cas No.197794-83-5
FormulaC31H53N9O6
SolubilitySoluble to 1 mg/ml in 20% acetonitrile / sterile water
Chemical Name(S,Z)-2-((Z)-((S)-2-((Z)-((2S,3R)-2-amino-1,3-dihydroxybutylidene)amino)-1-hydroxy-3-phenylpropylidene)amino)-N-((S,Z)-1-(((S)-5-guanidino-1-hydroxy-1-iminopentan-2-yl)imino)-1-hydroxy-4-methylpentan-2-yl)-4-methylpentanimidic acid
SDFDownload SDF
Canonical SMILESCC(C[[email protected]@](/N=C(O)/[[email protected]](/N=C(O)/[[email protected]](/N=C(O)/[[email protected]](N)([H])[[email protected]@](O)([H])C)([H])CC1=CC=CC=C1)([H])CC(C)C)([H])/C(O)=N/[[email protected]@](C(O)=N)([H])CCCNC(N)=N)C
Shipping ConditionEvaluation sample solution: ship with blue ice. All other available sizes: ship with RT, or blue ice upon request.
General tipsFor obtaining a higher solubility, please warm the tube at 37°C and shake it in the ultrasonic bath for a while. Stock solution can be stored below -20°C for several months.

Quality Control

Chemical structure

TFLLR-NH2