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TAK-700 (Orteronel)Human 17,20-lyase inhibitor

TAK-700 (Orteronel)

Catalog No. A4326
Size Price Stock Qty
10mM (in 1mL DMSO) $231.00 In stock
5mg $105.00 In stock
50mg $420.00 In stock

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Sample solution is provided at 25 µL, 10mM.

Product Citations

1. F. Peter Guengerich,Martin Egli,et al."The Kinetic and Chemical Mechanisms of Human Cytochrome P450 17A1." Vanderbilt University. 2017 May.

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Quality Control

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Chemical structure

TAK-700 (Orteronel)

Related Biological Data

TAK-700 (Orteronel)

TAK-700 (Orteronel) Dilution Calculator

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Chemical Properties

Cas No. 426219-18-3 SDF Download SDF
Chemical Name 6-(7-hydroxy-5,6-dihydropyrrolo[1,2-c]imidazol-7-yl)-N-methylnaphthalene-2-carboxamide
Canonical SMILES CNC(=O)C1=CC2=C(C=C1)C=C(C=C2)C3(CCN4C3=CN=C4)O
Formula C18H17N3O2 M.Wt 307.35
Solubility >11.2mg/mL in DMSO Storage Store at -20°C
General tips For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20℃ for several months.
Shipping Condition Evaluation sample solution : ship with blue ice
All other available size: ship with RT , or blue ice upon request

Background

TAK-700 (Orteronel) is a potent and highly selective human 17,20-lyase inhibitor with IC50 of 38 nM, exhibits >1000-fold selectivity over other CYPs (e.g. 11-hydroxylase and CYP3A4). Phase 3.