Search results for: 'research-area metabolism'
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- A3146 AGI-6780Target: IDH2Summary: IDH2/R140Q mutation inhibitor
- A4383 TolcaponeTarget: Catechol O-Methyltransferase (COMT)Summary: COMT inhibitor
- A4381 FK866 (APO866)1 CitationTarget: NamptSummary: NAMPT inhibitor, non-competitive, highly specific
- A4373 NLG9191 CitationSummary: Potent IDO pathway inhibitor
- A4365 LovastatinTarget: HMG-CoA ReductasesSummary: HMG-CoA reductase inhibitor
- A4358 U-104Target: Carbonic AnhydrasesSummary: CAIX inhibitor
- A4347 Methotrexate2 CitationTarget: Folate AnalogueSummary: Folate antagonist,inhibits DFHR
- A4346 AminophyllineTarget: Phosphodiesterases (PDEs)Summary: Pan-PDE inhibitor
- A4333 CPI-6131 CitationTarget: Pyruvate dehydrogenases (PDH)Summary: PDH/α-KGDH inhibitor
- A4330 IsotretinoinTarget: RARsSummary: Dopamine β-hydroxylase activator