Search results for: 'research-area mapk mapk-rasgap-ras-p21'
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- B2169 IPA-31 CitationTarget: PAKSummary: Non-ATP competitive Pak1 inhibitor
- B1162 FRAX5971 CitationTarget: PAKSummary: PAK inhibitor,potent and ATP-competitive
- A8501 PHA-848125Target: Cyclin-Dependent KinasesSummary: CDK inhibitor,potent and ATP-competitive
- A3716 PF-37583091 CitationTarget: PAKSummary: PAK4 inhibitor
- A4203 Tenovin-1Target: Sir2-like Family Deacetylases (Sirtuins)|p53|p21Summary: SIRT2 inhibitor, activates p53
- A3316 Clemizole hydrochlorideTarget: Histamine H1 Receptors|TRPC channelSummary: H1 histamine receptor antagonist
- B6012 Pexmetinib (ARRY-614)Target: p38|Tie-2Summary: dual inhibitor of p38 MAPK and Tie2/Tek receptor tyrosine kinase
- A5979 Tie2 kinase inhibitorTarget: Tie-2Summary: Tie-2(Tie2 ) inhibitor