Search results for: 'research-area gpcr-g-protein'
- Thioridazine HClCatalog No. :A8537Calcium channel protein inhibitorThioridazine·HCl is a calcium channel protein inhibitor as well as D2DR/D4DR inhibitor.
- I-CBP 112Catalog No. :A4490CBP/EP300 bromodomain inhibitorA bromodomain is an approximately 110 amino acid protein domain that recognizes monoacetylated lysine residues such as those on the N-terminal tails of histones.
- OTX-015Catalog No. :A3692BRD inhibitor
OTX-015 is a potent inhibitor of BRD2, BRD3, and BRD4 with IC50 values range from 92 to 112 nM
- PLX-4720Catalog No. :A3016BRAF kinase inhibitor
PLX-4720, a 7-azaindole derivative discovered by a structure-guided discovery approach, is a potent inhibitor of B-RafV600E, the most frequent oncogenic protein kinase mutation, with the value of 50% inhibition concentration IC50 of 13 nM.