Search results for: 'research-area gpcr-g-protein'
- Thioridazine HClCatalog No. :A8537Calcium channel protein inhibitorThioridazine·HCl is a calcium channel protein inhibitor as well as D2DR/D4DR inhibitor.
- I-CBP 112Catalog No. :A4490CBP/EP300 bromodomain inhibitorA bromodomain is an approximately 110 amino acid protein domain that recognizes monoacetylated lysine residues such as those on the N-terminal tails of histones.
- OTX-015Catalog No. :A3692BRD inhibitor
OTX-015 is a potent inhibitor of BRD2, BRD3, and BRD4 with IC50 values range from 92 to 112 nM
- Anacetrapib (MK-0859)Catalog No. :A4375RhCETP/mutant CETP(C13S) inhibitor
Anacetrapib, also known as MK-0859, is a potent and selective inhibitor of cholesteryl ester transfer protein (CETP) that exhibits strong inhibition against CETP-mediated transfer of cholesteryl esters and triglycerides with values of inhibition constant IC50 of 16 nM and 29 nM respectively.