Search results for: 'research-area gpcr-g-protein'
- Thioridazine HClCatalog No. :A8537Calcium channel protein inhibitorThioridazine·HCl is a calcium channel protein inhibitor as well as D2DR/D4DR inhibitor.
- KU-60019Catalog No. :A8336ATM kinase inhibitor,potent and selective
KU-60019 is a selective inhibitor of the Ataxia telangiectasia (A-T) mutated (ATM) protein with an IC50 value of 6.3 nM. In literature report, KU-60019 radiosensitizes h-TERT-immortalized normal fibroblasts but not A-T fibroblasts, suggesting it is a specific ATM kinase radiosensitizer .
- I-CBP 112Catalog No. :A4490CBP/EP300 bromodomain inhibitorA bromodomain is an approximately 110 amino acid protein domain that recognizes monoacetylated lysine residues such as those on the N-terminal tails of histones.
- OTX-015Catalog No. :A3692BRD inhibitor
OTX-015 is a potent inhibitor of BRD2, BRD3, and BRD4 with IC50 values range from 92 to 112 nM