Search results for: 'research area gpcr g protein glucocorticoid receptor'
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- A4064 NVP-BEP800Target: HSP90Summary: Oral Hsp90β inhibitor, novel, fully synthetic
- A3170 AM9662 CitationTarget: LPA ReceptorsSummary: LPA1 antagonist, oral active, high affinity, selective,
- B6342 H-7 dihydrochlorideTarget: PKC|PKG|PKA|Myosin light chain kinases (MLCKs)Summary: protein kinase inhibitor
- B1577 C6461 CitationTarget: p300Summary: HAT p300-CBP inhibitor,cell-permeable
- A3570 LY2090314Target: GSK-3Summary: Potent GSK-3 inhibitor
- A3347 Dabrafenib Mesylate (GSK-2118436)Target: RafSummary: Inhibitor of BRAF(V600) mutants
- A4388 XL-8881 CitationTarget: HSP90Summary: Hsp90 inhibitor
- B3278 BQ-788 sodium salt1 CitationTarget: Endothelin receptorsSummary: ET B-receptor antagonist,potent and selective
- A8370 Axitinib (AG 013736)1 CitationTarget: VEGFR|PDGFR|c-KitSummary: VEGFR1/ c-Kit inhibitor