Search results for: 'leu31-pro34-neuropeptide-y-human-rat'
- Ki16425Catalog No. :A1987LPA receptor antagonist
Ki16425 is a subtype-selective antagonist of lysophosphatidic acid receptor (LPA) with Ki values of 0.34 μM for LPA1, 6.5μM for LPA2, and 0.93μM for LPA3 .
- AM-095 free baseCatalog No. :A3167Potent LPA1 receptor antagonistAM095 is a novel, potent and orally bioavailable antagonist of lysophosphatidic acid type 1 receptor (LPA1) with IC50 values of 0.73 and 0.98 μM for mouse or recombinant human LPA1, respectively .
- AM966Catalog No. :A3170LPA1 antagonist, oral active, high affinity, selective,
AM966 is a selective, potent and orally bioavailable antagonist of lysophosphatidic acid type 1 receptor (LPA1) with IC50 values of 17 and 19 nM for human or mouse LPA1, respectively . Relative to LPA2, 3, 4, 5 receptors, AM966 shows 10-fold and 100-fold more selective in mouse and human cell lines for LPA1, respectively .