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DiscoveryProbe™ GPCR/G protein-related Compounds Panel

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A wide range of well-characterized bioactive molecules that covers various targets related to GPCR, including adenosine receptor, adrenergic receptor and CXCR etc. Facilitate your research towards the insights of cancer, neurological disorders and heart diseases etc. Applicable in cellular assays, animal models and drug screenings etc.

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Related Biological Data


Related Biological Data



Available in stock with overnight delivery and free shipping over $500 Cost-effective and competitive price to save your findings Potent, selective and cell-permeable in inhibiting or activating target molecules Diverse in chemical structure and route of administration (oral/i.m/i.v injection etc.) Detailed files describing potency, selectivity and applications etc. Supported by published data from top peer-reviewed journals Guaranteed high quality with NMR and HPLC validation

Featured Products of the Panel

Catalog No. Product Name Summary Targets CAS Number Smiles
A8454 Istradefylline (KW-6002) Selective A2A receptor antagonist GPCR/G protein|Adenosine Receptor 155270-99-8 CCN1C2=C(C(=O)N(C1=O)CC)N(C(=N2)C=CC3=CC(=C(C=C3)OC)OC)C
B1007 AVE 0991 Agonist of angiotensin-(1-7) receptor GPCR/G protein|Angiotensin Receptor 304462-19-9 CCNC(=O)NS(=O)(=O)C1=C(C=C(S1)CC(C)C)C2=CC=C(C=C2)CN3C(=C(N=C3C4=CC=CC=C4)OC)C=O
A1435 CP-945598 HCl CB1 antagonist,selective and high affinity GPCR/G protein|Cannabinoid Receptor 686347-12-6 CCNC1(CCN(CC1)C2=NC=NC3=C2N=C(N3C4=CC=C(C=C4)Cl)C5=CC=CC=C5Cl)C(=O)N.Cl
A5827 AM1241 Cannabinoid CB2 receptor agonist,potent and selective GPCR/G protein|Cannabinoid Receptor 444912-48-5 CN1CCCCC1CN2C=C(C3=CC=CC=C32)C(=O)C4=C(C=CC(=C4)[N+](=O)[O-])I
A2025 Plerixafor (AMD3100) CXCR4 antagonist; CXCR7 agonist GPCR/G protein|CXCR 110078-46-1 C1CNCCNCCCN(CCNC1)CC2=CC=C(C=C2)CN3CCCNCCNCCCNCC3
A3802 SCH 527123 CXCR1 and CXCR2 receptors antagonist GPCR/G protein|CXCR 473727-83-2 CCC(C1=CC=C(O1)C)NC2=C(C(=O)C2=O)NC3=CC=CC(=C3O)C(=O)N(C)C
B1633 CTEP (RO4956371) MGlu5 inhibitor GPCR/G protein|mGluR 871362-31-1 CC1=C(N=C(N1C2=CC=C(C=C2)OC(F)(F)F)C)C#CC3=CC(=NC=C3)Cl
A3616 MK-4305 OX1/OX2 atagonist,potent and selective GPCR/G protein|OX Receptor 1030377-33-3 CC1CCN(CCN1C(=O)C2=C(C=CC(=C2)C)N3N=CC=N3)C4=NC5=C(O4)C=CC(=C5)Cl
B2166 Ticagrelor P2Y12 receptor antagonist GPCR/G protein|P2Y Receptor 274693-27-5 CCCSC1=NC2=C(C(=N1)NC3CC3C4=CC(=C(C=C4)F)F)N=NN2C5CC(C(C5O)O)OCCO
Download the GPCR/G protein-related Compounds Panel - XLSX       Download the GPCR/G protein-related Compounds Panel - SDF


1. Wettschureck N, Offermanns S. Mammalian G proteins and their cell type specific functions. Physiol Rev. 2005 Oct;85(4):1159-204.
G protein-mediated signaling is employed by virtually all cells in the mammalian organism and is centrally involved in diverse physiological functions such as perception of sensory information, modulation of synaptic transmission, hormone release and actions, regulation of cell contraction and migration, or cell growth and differentiation. In this review, some of the functions of heterotrimeric G proteins in defined cells and tissues are described.